CV
CURRIUCULUM VITA
Ayman Ahmed El-Faham
E-mail: aelfaham@ksu.edu.sa; aymanel_faham@hotmail.com.; http://fac.ksu.edu.sa/aelfaham
web of science h-index 31, citation 4516; Google Scholar h-index 37, citation 6384;
Scopus 31, citation 4609
ORCID ID; 0000-0002-3951-2754; Scopus ID: 7004414569: 35315447500;
ResearcherID: G-1554-2010
https://scholar.google.com/citations?user=iPCDQWwAAAAJ&hl=en
RESEARCH INTEREST
Professor of Organic Chemistry focuses on the synthesis and characterization of peptides, peptide coupling reagents, green chemistry and microwave synthesis of biologically active compounds.
Personal Data
Date of Birth: April 7th, 1958
Place of Birth: Alexandria, Egypt.
Current Address:
King Saud University, College of Science, Chemistry Department
P.O. Box 2455, Riyadh 11451, Saudi Arabia
Tel: 0096616473195. Mobile: 00966544871738.
Permanent Address:
Work address:
Alexandria University, Faculty of Science, Chemistry Department
P.O. Box426, Ibrahimia, 21321 Alexandria, Egypt.
Tel: 00203-5922352.
QUALIFICATIONS & AWARDS
- Unilever Sustainable Living Plan Prize for the best Article (2016).
- Award of Excellence in Scientific Publishing from Quality Authority (CIQAP) Egypt (2012).
- Prize of Administrative Excellence Alexandria University 2012.
- Medal for Distinguish Scientific Publication in Chemistry, Alexandria University (2010)
- Invited to submit a proposal for Noble Prize in Chemistry (2003)
- Alexandria University Award for Science 1999 (In Chemistry)
- Prof. Abd El-Fatah Ismail Award for highest achieving student in Faculty of Science, Alexandria University, Egypt, (1980)
- 201 publications, 45 conferences papers, 4 book chapters, 12 US Patents, and 1 Egyptian Patent.
EDUCATION
D. Sc., 2010: Faculty of Science, Chemistry Department, Alexandria University, Alexandria-Egypt. “Peptide Synthesis"
Ph. D., 1991: University of Massachusetts, U. S. A. and University of Alexandria, Egypt
(Joint Supervision) “The 9-Fluorenylmethyl Function as a potential Amino-Protecting Group in Peptide Synthesis”
M. Sc., 1985: Faculty of Science, Chemistry Department, Alexandria University, Alexandria- Egypt “Kinetic and Mechanism of the Action of Alkalis on Nitro-diphenylmethyl Thio-Compounds”
B. Sc., 1980: Faculty of Science, Chemistry Department, Alexandria University, Alexandria-Egypt.
Scholaeships and Sabbaticals
- 10/2011-now. Professor, King Saud University, College of Science, Chemistry Department, Saudi Arabia, Riyadh.
- 2010 – 2011. Vice-Dean for Community Development & Environmental Affairs, University of Alexandria, Faculty of Science, Alexandria-Egypt.
- 07/2011-09/2011. Visiting Professor, University of Barcelona (Barcelona Science Park) Barcelona, Spain.
- 2008- 2010. Professor of Organic Chemistry, King Saud University, College of Science, Chemistry Department, Saudi Arabia, Riyadh.
- 07/2009-09/2009. Visiting Professor, University of Barcelona, Department of Chemistry, Barcelona, Spain.
- 2004- 2008. Direct Manager of the Central Lab and NMR Lab (Nuclear Magnetic Resonance Lab).Alexandria University, Faculty of Science, Chemistry Department, Alexandria, Egypt.
- 07/2008-09/2008. Visiting Professor, University of Barcelona (Barcelona Science Park), Barcelona, Spain.
- 06/2007-09/2007. Visiting Professor, University of Barcelona (Barcelona Science Park), Barcelona, Spain.
- 06/2006-09/2006. Visiting Professor, University of Barcelona (Barcelona Science Park) Barcelona, Spain.
- 2000- 2004. Head of the Chemistry Department, Beirut Arab University, Faculty of Science, Beirut, Lebanon.
- 07/1999-10/1999. Visiting Professor, University of Massachusetts, Department of Chemistry, Amherst, MA 01003, U. S. A.
- 1996-1998. Post-Doctoral Research Associate, University of Massachusetts, Department of Chemistry, Amherst, MA 01003, U. S. A.
- 07/1995-10/1995. Visiting Professor, University of Massachusetts, Department of Chemistry, Amherst, MA 01003, U. S. A.
- 1992-1994. Post-Doctoral Research Associate, University of Massachusetts, Chemistry Department, Amherst, MA 01003, U. S. A.
- 1989-1991. Research Assistant, University of Massachusetts, Chemistry Department, Amherst, MA 01003, U. S. A., and Ph. D. dissertation research.
- 1986-1989. Research Assistant, University of Alexandria, Chemistry Department, Faculty of Science, Alexandria-Egypt, Ph. D. dissertation research.
- 1980-1986. Research Assistant, University of Alexandria, Chemistry Department, Faculty of Science, Alexandria-Egypt, M. Sc. dissertation research.
Funded Projects
- CO-PI: King Abdul-Aziz city for Science and Technology (KACST). Synthesis and Study Novel Co-Polymers Based on s-Triazine Unit and its Ability in Ion Extraction upon Complexation Technique" 2016-2017.
- PI: King Abdul-Aziz city for Science and Technology (KACST), Saudi Arabia project No. (SGP-34-55) "Synthesis and Biological Screening of Novel Series of Isatin-Triazine Derivatives. 2014-2015.
- CO-PI: Science and Technology Development Fund (STDF) funded project. Coupling Reagents: Applications in Solution and Solid-Phase. Synthesis of Biologically Active Peptide. 2012-2013.
- PI: King Saud University, Deanship of Scientific Research, College of Science Research Center (Chem/2010/02). Easy way for the synntesis of Novel thino[2,3-b]thinophene derivatives. 2010- 2011.
- CO-PI: King Saud University, Deanship of Scientific Research, College of Science Research Center (Chem/2010/02). Solventless Microwave Synthesis of Biologically active amino acid hydrazide-hydrazone derivatives as a promosing technique for development antimicrobial agents” 2010- 2011.
- PI: Agencia Espanola De Cooperacion Internacional (AECI) “Reactivos Para La Sintesis De Peptidos Con Actividad Terapeutica" 2008- 2009.
- PI: Beirut Arab University Collaboration with Dubai. Bioremediation of Industrial Waste Water by Marine Algae. 2003-2006.
- PI: Conseil National De La Recherche Scientifique, Lebanon (CNRS). Design and Synthesis of Novel Coupling Regeants Used in Synthesis of Biological Active Peptides. 2003-2004.
Training Course and Workshops
- Course Specification and Report (King Saud University, Saudi Arabia,02-03/2/2016)
- Critical thinking and active Learning (King Saud University, Saudi Arabia,09-10/09/2015)
- Collaboration between the Universities and Privet Sector in Scientific Research (King Saud University, Saudi Arabia 28-19/10/2015)
- 3rd International Symposium on Chemical and Biological Safety and Training Workshops, King Saud University, Saudi Arabia (May12-14, 2015)
- Usage of Smart Classrooms (22/12/2012, 5 hours, King Saud University, Saudi Arabia.
- Recent Trends in Learning Technology (2-3/9/2012) King Saud University, Saudi Arabia.
- Basic of Electronic Learning Management System (4-5/9/2012) King Saud University, Saudi Arabia.
- Learning Outcomes and Curriculum Maps (32 hours18-22/12/2010).
- External Review of Higher Education Institutions (32 hours, 18-22/9/2010).
- Practice and Documents Supporting Self-Study (32 hours, 7-11/8/2010). University of Alexandria, Faculty of Science, Alexandria, Egypt.
- The Self Study Practice and Documents Required for High Education (12 hours, 26- 27/7/2010).University of Alexandria, Faculty of Science, Alexandria, Egypt.
- DNA Research: A Gateway to the Knowledge Economy (24/5/2009) King Saud University, Saudi Arabia.
- Course Development (25-27/10/2008, 12 hours) King Saud University, Saudi Arabia.
- Quality Control and Assurance for Chemical Analysis (16-18/3/2008, 20 hours). City for Scientific Researcher and Technology, Alexandria, Egypt.
- Nuclear Magnetic Resonance (NMR-ECA-500) Applications JEOL Ltd. Japan.
Supervised Theses
- 14 Ph.D. Thesis; 17 M.Sc. Thesis
Professional Skills
- 40 years of bench research experience in Synthetic Organic, Peptide, Glycopeptide, Combinatorial Chemistry and Heterocyclic Chemistry.
- Hands-on skills in multi-step Organic Synthesis, Solid and Solution-Phase Organic and Peptide Synthesis, Microwave synthesis. Synthesis of peptides using a large variety of protecting groups, coupling reagents and additives in solution and solid phase techniques, heterocyclic synthesis, and polymer synthesis.
- Use of modern physical methods (1H, 13C, High Field NMR, MS. FT-IR, HPLC, GC-MS, UV, TLC, etc.) in the monitoring of chemical reactions, purification and characterization of products, mechanistic approach of organic reactions using physical methods (NMR, IR, UV, HLPC) by isolation and characterization of some intermediates
- Working from laboratory to pilot-plant scales with air/moisture sensitive, inflammable and poison reagents at normal-/or under vacuum.
- Very good experiences in dealing with computer and new teaching programs, molecular modeling.
TEACHING Experiences
- 2011-now, Professor of Organic Chemistry and Peptides, King Saud University, College of Science, Chemistry Department, Saudi Arabia, Riyadh.
- 2008- 2010, Professor of Organic Chemistry, King Saud University, College of Science, Chemistry Department, Saudi Arabia, Riyadh.
- 2004 - 2008, Professor of Organic Chemistry and Peptides, University of Alexandria, Faculty of Science, Chemistry Department, Alexandria-Egypt.
- 2000 –2004, Professor of Organic Chemistry and Peptides, Beirut Arab University, Faculty of Science, Chemistry Department, Beirut, Lebanon.
- 1996 - 2000, Associate Professor in Organic Chemistry and Peptides, University of Alexandria, Faculty of Science, Chemistry Department, Alexandria-Egypt.
- 1991-1996, Lecturer in Organic Chemistry, Alexandria University, Faculty of Science, Chemistry Department, Alexandria-Egypt.
- 1985-1991, Assistant Lecturer in Physical Organic Chemistry, Alexandria University, Faculty of Science, Chemistry Department, Alexandria-Egypt.
- 1980-1985, Demonstrator in Chemistry, Alexandria University, Faculty of Science, Chemistry Department, Alexandria-Egypt
Other Community - University Activities
- 2010-2012, Member of the Research Scientific Committee, Alexandria University.
- Supervisor of the incubating graduate project program, King Saud University“2008-2010”
- Direct Manager of the Central Lab. Unit and NMR lab, Faculty of Science, Alexandria University "Consulting Advices - Analytical performances - IR, UV-VIS, EA, GC-MS, HPLC and NMR Spectroscopy "2004-2008”.
- Direct Manager of the Central Lab. Unit, Moubark City for Applied Research and Technology, Borg Alarab, Alexandria ¨2007-2008”.
- Direct Manager of the Central Lab. Unit, Beirut Arab University, Faculty of Science, Chemistry Department, Lebanon "Consulting Advices - Analytical performances - IR, UV-VIS, EA, GC-MS, HPLC and NMR Spectroscopy " 2000-2004.
- Member of the organizing committee for international contacts "The 7 th
- Ibn Sina International Conference on pure and applied heterocyclic Chemistry" (7 th
- ISCHC), 25-28 th March 2000, Alexandria, EGYPT.
- Faculty of Science Alumni Association – Alexandria University, Member "Consulting Advices - Analytical performances".
- Scientific Chemical Association – Faculty of Science – Alexandria University, Member "Organizing and giving seminars on Modern Chemistry"
- Head of different groups of the student union activities over about 20 years.
Editorial Activities
- Pre-reviewer for the Chemistry Program (B.Sc.), Al Amam Mohammed Bin Saud Islamic University, Saudi Arabia. Since 2019.
- A member of the Board of Directors of Saudi Chemical Society since 2013-2016.
- The Saudi Chemical Society since 2013.
- Member of the American Chemical Society since 2008.
- Member of the Arab Society of Material Science since 1991.
- Member of the Egyptian Heterocyclic Society since 1991.
- Faculty of Science Alumni Association.
- Academic editor Journal of Molecular Pharmaceutics & Organic Process Research since 2013.
- Member of Editorial Board for Journal of Green and Sustainable chemistry since 2010.
- Academic Editor International Journal of Peptide Science (Int.J.Pept.Sci) since 2008.
- Member of Editorial Board for Saudi Journal of Chemical Society (SJCS) since 2008
- Reviewer for Tetrahedron since 2008.
- Member of Editorial Board for Saudi Chemical Society since 2009.
- Editorial Board Referee for ARKIVOC (USA) journal since 2003.
- ACS Chemistry Ambassador since 2015.
- Academic Member of the Athens Institute for Education and Research since 2015
- Member of BIT since 2016.
List of Publications
I- US Patents.
- Ayman El-Faham, Zeid ALOthman, Sameh Osman. Modification of methoxy polyethylene glycol for synthesis of metal nanoparticles in liquid and solid phase” U.S. Patent 9,873,153 B1; Jan, 23, 2018.
- Ayman El-Faham, Moustafa M. G. E. Fouda, Zeid A. ALOthman. Functionalized silica for the synthesis of metal nanoparticles US Patent 9,636,747 B1, 2 May 2017.
- Kareem Y. H. Mahmoud, Zeid A. ALOthman, Ayman El-Faham. Functionalizable monolithic platforms. US Patent 9,624,335 B1, 18 April 2017.
- Sherine A. N. Khattab, Ayman El-Faham, Mona I. Massoud, Yahya E. Jad. Production of new sweeteners from stevioside extracted from stevia plant. WO 27066, 2015 (Egyptian Patent).
- Fernando Albericio, Ayman El-Faham, et al. New Oxime Coupling Agent Useful in Preparing Polynucleotide and Peptide. US Patent, (2009) WO2009138985-A2.
- Fernando Albericio, Ayman El-Faham. Proton Acceptor Immonium-type Coupling Reagents. US Patent (2008) 20-11-2008, WO2008/139481-A2, WO2008139481-A3.
- L. A. Carpino, H. Imazumi,and Ayman El-Faham"New cationic portion of uranium or immonium salts useful for carrying out acylation step in amide formation, particularly during peptide synthesis" US Patent WO200294822-A; -A1; US 2003125561-A1; EP 1395584-A1; AU2002310004-A1; US6825347-B2; JP2005500268-W; AU2002310004-B2, 2003.
- L. A. Carpino, H. Imazumi,and Ayman El-Faham. New 2-Heterocyclyl-Pyridine 1-oxide Derivatives Useful as Herbicides for Pre-and Post-emergence Weed Control” US Patent WO200294822-A; WO200294822-A1; US2003125561-A1.
- L. A. Carpino, H. Imazumi,and Ayman El-Faham “ New Peptide Coupling Reagents: The Authentic Uronium Salt” US Patent no.6,825,347, Nov. 30, 2004.
- L. A. Carpino and Ayman El-Faham “Synthesis and Use of Amino Acid Fluorides as Peptide Coupling Reagents” US Patent no. 6, 534, 627, March 18, 2003.
- L. A. Carpino and Ayman El-Faham “Synthesis and Use of Amino Acid Fluorides as Peptide Coupling Reagents” US Patent no. 6, 040, 422, March 21, 2000.
- L. A. Carpino and Ayman El-Faham “Synthesis and Use of Amino Acid Fluorides as Peptide Coupling Reagents” US Patent no. 5,712,418, May 12, 1998.
- L. A. Carpino and Ayman El-Faham “Synthesis and Use of Amino Acid Fluorides as Peptide Coupling Reagents” US Patent no. 5,750,767, January 27, 1998.
II- Chapter in Books
- Y. Jad, Ayman El-Faham, B. G. de la Torre, and F. Albericio” Solid-Phase Peptide Synthesis, the State of the Art: Challenges and Opportunities” Peptide-based Drug Discovery: Challenges and New Therapeutics., Royal Society of Chemistry, Chapter 18, (2017), pp 515-550, Print ISBN 978-1-7826-732-6.
- J. Tulla-Puche, Ayman El-Faham, A. S. Galanis, E. de Oliveira, A. A. Zompra, and F. Albericio “Peptide Drugs: Peptide Chemistry and Drug Design : Chapter 4. ‘Methods for the Synthesis and Analysis of Peptides” (Ben M. Dunn, ed.) Wiley Sons, (2015) pp 11- 73.
- Ayman El-Faham and Fernando Albericio “Amino Acids, Peptides and Proteins in Organic Chemistry, Vol. 3-Building Blocks, Catalysis and Coupling Chemistry (Andrew B. Hughes, Ed.) Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim (Germany), Chapter 12, (2011) pp 407-446.
- Ayman El-Faham, Ramon Subiros-Funosas and Fernando Albericio “N-Hydroxyamines for peptide synthesis”. In The chemistry of hydroxylamine, oxime and hydroxamic acid, Volume 2 (Z. Rappoport and J. F. Liebman eds.) Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim (Germany), Chapter 11 (2011) pp 623-730
III-Publications
- A. Barakat, S. M. Soliman, M. Ali, A. Elmarghany, A. M. Al-Majid, S. Yousuf, Z.Ul-Haq, M. I. Choudhary, Ayman El-Faham. Synthesis, crystal structure, evaluation of urease inhibition potential and the docking studies of cobalt(III) complex based on barbituric acid Schiff base ligand. Inorganic Chimica Acta, In press 2020; doi.org/10.1016/j.ica.2019.119405
- H. H. Al-Rasheed, S. Z. Mohammady, Kh. Dahlous, M. R. H. Siddiqui, Ayman El-Faham. Synthesis, characterization, thermal stability and kinetics of thermal degradation of novel polymers based-s-triazine Schiff base. Journal of Polymer Research, (2020) 27:10, 1-11; doi.org/10.1007/s10965-019-1961-8
- Ayman El-Faham, M. Farooq, Z. Almarhoon, R. Abd Alhameed, M. A. M. Wadaan, B. G. de la Torre, F. Albericio. Di- and tri-substituted s-triazine derivatives: Synthesis, characterization, anticancer activity in human breast-cancer cell lines, and developmental toxicity in zebrafish embryos. Bioorg. Chem. 94 (2020) 103397 doi: 10.1016/j.bioorg.2019.103397
- Barakat , S. M. Soliman, Ayman El-Faham, M. Ali, A. M. Al-Majid, S. Yousuf, M. I. Choudhary. Three Multi-Components Reaction: Synthesis and X-Ray Single-Crystal of Hydroacridinone-Based Hydrazino-S-Triazine Derivative as a New Class of Urease Inhibitor. Crystals 2020, 10, 14; doi:10.3390/cryst10010014.
- R. Abd Alhameed, Z. Almarhoon, S. I. Bukhari, Ayman El-Faham, B. G. de la Torre, F. Albericio. Synthesis and Antimicrobial Activity of a New Series of Thiazolidine-2,4-diones Carboxamide and Amino Acid Derivatives. Molecules 2020, 25, 105; doi:10.3390/molecules25010105.
- S. M. Soliman, J. Lasri, M. Haukka, E. N. Sholkamy, H. H. Al-Rasheed, Ayman El-Faham. Synthesis, X-ray Crystal Structure and Antimicrobial Activity of Unexpected Trinuclear Cu(II) Complex from s-Triazine-Based Di-Compartmental Ligand via Self-Assembly. Crystals 2019, 9, 661; doi:10.3390/cryst9120661
- Z. Almarhoon, Kh. A. Dahlous, R. Abd Alhameed, H.A. Ghabbour, Ayman El-Faham. A Simple, Efficient, and Eco-Friendly Method for the Preparation of 3-Substituted-2,3-dihydroquinazolin-4(1H)-one Derivatives. Molecules 2019, 24, 4052; doi:10.3390/molecules24224052
- A. Sharma, R.Sheyi, A. Kumar, Ayman El-Faham, B.G. de la Torre, and Fernando Albericio. Investigating Triorthogonal Chemoselectivity. Effect of Azide Substitution on the Triazine Core. Org. Lett. 2019, 21, 2459−2463; doi: 10.1021/acs.orglett.9b02878
- O. Al Musaimi, Ayman El-Faham, A. Basso, B. G. de la Torre, F. Albericio. γ-Valerolactone (GVL): An eco-friendly anchoring solvent for solid-phase peptide synthesis. Tetrahedron Letters, 2019, 60, 151058; doi: 10.1016/j.tetlet.2019.151058
- S. M. Soliman, Z. Almarhoon, E. N. Sholkamy, Ayman El-Faham. Bis-pyrazolyl-s-triazine Ni(II) pincer complexes as selective gram positive antibacterial agents; synthesis, structural and antimicrobial studies. J. Mol. Str. 2019, 1195, 315-322; doi: 10.1016/j.molstruc.2019.05.103.
- A. ur R. Khan, M. Nadeem, M. Aqeel Bhutto, F.Yu, X. Xie, H. El-Hamshary, Ayman El-Faham, U.A. Ibrahim and X. Mo. Physico Chemical and Biological Evaluation of PLCL/SF Nanofibers Loaded with Oregano Essential Oil. Pharmaceutics 2019, 11, 386 (1-18); doi:10.3390/pharmaceutics11080386.
- D. Carbajo, P. Fransen, Ayman El-Faham, M. Royo, and F. Albericio. Pseudo-Wang Handle for the Preparation of Fully Protected Peptides. Synthesis of Liraglutide by Fragment Condensation. Org. Lett. 2019, 21, 2459−2463; doi: 10.1021/acs.orglett.9b00813.
- D. Carbajo, Ayman El-Faham, M. Royo, and F. Albericio. Optimized Stepwise Synthesis of the API Liraglutide Using BAL Resin and Pseudoprolines. ACS Omega 2019, 4, 8674−8680; doi: 10.1021/acsomega.9b00974.
- S. M. Soliman, Ayman El-Faham. Synthesis, X-ray structure and DFT studies of five- and eight-coordinated Cd(II) complexes with s-triazine N-pincer chelate. J. Coord. Chem., 2019, 72, 1621-1636; doi: 10.1080/00958972.2019.1608360.
- S. M. Soliman, Ayman El-Faham, J. Albering. Cu(II)-promoted cyclization of Hydrazonophthalazine to triazolophthalazine; Synthesis and structure diversity of six novel copper(II) complexes. Applied Organometallic Chemistry; 2019; e4992; doi.org/10.1002/aoc.4992.
- S. M. Soliman, Z. Almarhoon and Ayman El-Faham. Synthesis, Molecular and Supramolecular Structures of New Cd(II) Pincer-Type Complexes with s- Triazine Core Ligand. Crystals 2019, 9, 226 (1-16); doi:10.3390/cryst9050226.
- Othman Al Musaimi, Ayman El-Faham, Zainab Almarhoon, Alessandra Basso, Beatriz G. de la Torre, and Fernando Albericio. Bypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective. Polymers 2019, 11, 874 (1-13) ; doi:10.3390/polym11050874.
- A. Barakat, Fardous F. El-Senduny, Z. Almarhoon, H. H. Al-Rasheed, F. A. Badria, A. M. Al-Majid, H. A. Ghabbour, and Ayman El-Faham. Synthesis, X-Ray Crystal Structures, and Preliminary Anti-proliferative Activities of News-Triazine-hydroxybenzylidene Hydrazone Derivatives. Journal of Chemistry 2019, Volume 2019, Article ID 9403908, 10 pages ; doi: 10.1155/2019/9403908.
- A. Sharma, Z. M. Almarhoon, Ayman El-Faham, B. G. de la Torre and F. Albericio. Efficient Route for Synthesis of Enamines from 1,3-Alkyl-2-Thioxodihydropyrimidine-4,6(1H,5H)-dione Enols. Lett. in Org. Chem., 2019, 16, 538-540; doi: 10.2174/1570178616666190409145118
- S. M. Soliman, Ayman El-Faham "Synthesis and structural DFT studies of Ni(II) and Co(II) complexes with s-triazine-based di-compartmental ligand" Polyhedron 2019, 165, 162–170; doi: 10.1016/j.poly.2019.03.024
- S. M. Soliman, Ayman El-Faham. Synthesis, molecular structure and DFT studies of two heteroleptic nickel(II) s-triazine pincer type complexes. J. Mol. Str., 2019, 1185, 461-468; doi: 10.1016/j.molstruc.2019.02.089
- M. Farooq, A. Sharma, Z. Almarhoon, A. Al-Dhfyan, Ayman El-Faham, N.Abu Taha, M. A. M. Wadaan, B. G. de laTorre, F. Albericio. Design and synthesis of mono-and di-pyrazolyl-s-triazine derivatives, their anticancer profile in human cancer cell lines, and in vivo toxicity in zebrafish embryos. Bioorg. Chem., 2019, 87, 457–464; doi: 10.1016/j.bioorg.2019.03.063.
- Y. E. Jad, A. Kumar, Ayman El-Faham, B. G. de la Torre, F. Albericio. Green Transformation of Solid-Phase Peptide Synthesis. ACS Sustainable Chem. Eng., 2019, 7, 3671−3683. doi: 10.1021/acssuschemeng.8b06520.
- D. Carbajo, Peter Fransen, Ayman El-Faham, M. Royo, F. Albericio. Pseudo-Wang Handle for the Preparation of Fully Protected Peptides. Synthesis of Liraglutide by Fragment Condensation. Org. Lett. 2019, 21, 2459−2463; doi: 10.1021/acs.orglett.9b00813.
- S. M. Soliman, Ayman El-Faham. Synthesis and structure diversity of high coordination number Cd(II) complexes of large s-triazine bis-Schiff base pincer chelate. Inorganica Chimica Acta 2019, 488, 131–140; doi: 10.1016/j.ica.2019.01.018.
- S. A. H. Abdel Monaim, A. M. Somboro, Ayman El-Faham, B. G de la Torre, F. Albericio. Bacteria Hunt Bacteria through an Intriguing Cyclic Peptide. ChemMedChem, 2019, 14, 24 – 5; doi: 10.1002/cmdc.201800597.
- Z. Almarhoon, S. M. Soliman, H. A. Ghabbour, Ayman El-Faham. A Facile and Eco-Friendly Method for the Synthesis of Sulfonamide and Sulfonate Carboxylic Acid Derivatives—X-ray Structure, Hirshfeld Analysis and Spectroscopic Characterizations. Crystals 2019, 9, 35; doi:10.3390/cryst9010035.
- H. El-Hamshary, M. H. El-Newehy, M.M. Abdulhameed, Ayman El-Faham, A. S. Elsherbiny . Evaluation of clay-ionene nanocomposite carriers for controlled drug delivery: Synthesis, in vitro drug release, and kinetics. Mater. Chem. Phy., 2019, 225, 122–132; dio: 10.1016/j.matchemphys.2018.12.054.
- K. A. Dahlous, O.H. Abd-Elkader, M.M.G. Fouda, Z.A. ALOthman, Ayman El-Faham. Eco-friendly method for silver nanoparticles immobilized decorated silica: Synthesis & characterization and preliminary antibacterial activity. J. Taiwan Inst. Chem. Eng., 2019, 95,423-331; doi.org/10.1016/j.jtice.2018.07.020.
- A. Sharma, Ayman El-Faham, B. G. de la Torre, F. Albericio. Exploring the Orthogonal Chemoselectivity of 2,4,6-Trichloro-1,3,5-triazine (TCT) as a Trifunctional Linker with Different Nucleophiles: Rules of the Game" Frontiers Chem.,2018, 6, 516. doi: 10.3389/fchem.2018.00516.
- O. Al Musaimi, Y. E. Jad, A. Kumar, Ayman El-Faham, J. M. Collins, A. Basso, B. G de la Torre, F. Albericio. Greening the Solid-Phase Peptide Synthesis Process. 2-MeTHF for the Incorporation of the First Amino Acid and Precipitation of Peptides after Global Deprotection. Org. Process Res. Dev., 2018, 22 (12), 1809–1816; doi: 10.1021/acs.oprd.8b00335.
- A. Sharma, S. J. Zamisa, S. Noki, Z. Almarhoon, Ayman El-Faham, B.G. de la Torre, F. Albericio. Crystal structure, spectroscopic studies and theoretical studies of thiobarbituric acid derivatives: understanding the hydrogen-bonding patterns. Acta Cryst. 2018, C74, 1703-1714; doi: 10.1107/S2053229618015516.
- K. A. Dahlous, Z. Almarhoon, A.-Y. B.-H.-Ahmed, Z. A. AL Othman, Ayman El-Faham. Microwave Irradiation Assists the Synthesis of a Novel Series of bis-Arm s-Triazine Oxy-Schiff Base and Oxybenzylidene Barbiturate Derivatives. Molecules 2018, 23, 2976; doi:10.3390/molecules23112976 (1-13).
- E. Kenawy, S. M. Osman, Z. A AlOthman, E. A. Aly, S. N. Khattab, Ayman El-Faham. Nitrogen containing polymers-based triazine: Synthesis, Characterization and its applications for scavenging of copper(II)" Desalination and Water Treatment, 2018, 114, 242–250; doi: 10.5004/dwt.2018.22386.
- Ayman El-Faham, A. M Atta, S.M Osman, A.O. Ezzat, A. M. El-Saeed, Z. A. A. L. Othman, H. A. Al-Lohedan. Silver-embedded epoxy nanocomposites as organic coatings for steel. Prog. Org. Coatings, 2018, 123, 209-222; doi: 10.1016/j.porgcoat.2018.07.006.
- A. M. Atta, Ayman El-Faham, H. A. Al-Lohedan, Z. A. AL Othman, M. M.S. Abdullah, A. O. Ezzat. Modified triazine decorated with Fe3O4 and Ag/Ag2O nanoparticles for self-healing of steel epoxy coatings in seawater. Prog.Org. Coatings, 2018, 121, 247-262; doi.org/10.1016/j.porgcoat.2018.04.011.
- S. M. Soliman, Ayman El-Faham. One pot synthesis of two Mn (II) perchlorate complexes with s-triazine NNN-pincer ligand; molecular structure, Hirshfeld analysis and DFT studies. J. Mol. Str., 2018, 1164, 344-353; doi.org/10.1016/j.molstruc.2018.03.037.
- A. Sharma, S. Noki, S.J. Zamisa, H.A. Hazzah, Z.M. Almarhoon, Ayman El‐Faham, G. Beatriz, F. Albericio. Exploiting the Thiobarbituric Acid Scaffold for Antibacterial Activity" ChemMedChem, 2018, 13, 1–9; doi: 10.1002/cmdc.201800414.
- S. M. Soliman, Ayman El-Faham, S. E. Elsilk, M. Farooq. Two heptacoordinated manganese (II) complexes of giant pentadentate s-triazine bis-Schiff base ligand: Synthesis, crystal structure, biological and DFT studies. Inorganica Chimica Acta, 2018, 479, 275-285; doi.org/10.1016/j.ica.2018.04.043.
- F. Albericio, Ayman El-Faham. Choosing the Right Coupling Reagent for Peptides. A Twenty-Five-Year Journey. Org. Process Res. Dev. 2018, 22, 760−772, doi: 10.1021/acs.oprd.8b00159.
- S. A. H. Abdel Monaim, J. T. Mhlongo, A. Kumar, Ayman El-Faham, F. Albericio, B. G. de la Torre" Formation of N-alpha-terminal 2-dialkyl amino oxazoles from guanidinated derivatives under mild conditions" Org. Biomol. Chem, 2018, 16, 5661-5666; doi: 10.1039/c8ob01463a
- S. M. Soliman, Ayman El-Faham "Synthesis, characterization and structural studies of two heteroleptic Mn(II) complexes with tridentate N,N,N-pincer type ligand. J. Coord. Chem., 2018, 1-16, doi: 10.1080/00958972.2018.1475660.
- M. A.M. Abu-Youssef, S. M. Soliman, Ayman El-Faham, J. Albering, M.M. Sharaf. A new triazoloquinoxaline ligand and its polymeric 1D silver (i) complex: synthesis, structure, and antimicrobial activity. New J. Chem., 2018, 42 (9), 7197-7205; doi: 10.1039/C7NJ02886E.
- S.A.H.A. Monaim, Y.E. Jad, Ayman El-Faham, B. G. de la Torre, F. Albericio. Teixobactin as a scaffold for unlimited new antimicrobial peptides: SAR study. Bioorg. Med. Chem., 2018, 26 (10), 2788-2796; doi.org/10.1016/j.bmc.2017.09.040.
- Sh. A.H. Abdel Monaim, G. A. Acosta, M. Royo, Ayman El-Faham, B.G. de la Torre, F. Albericio. Solid-phase synthesis of homodetic cyclic peptides from Fmoc-MeDbz-resin. Tetrahedron Lett., 2018, 59(18), pp. 1779-1782; doi.org/10.1016/j.tetlet.2018.03.084.
- Sh. N. Khattab, H. H. Khalil, A. A. Bekhit, M. M. Abd El-Rahman, B. G. de la Torre, Ayman El-Faham, and F. Albericio. 1,3,5-Triazino Peptide Derivatives: Synthesis, Characterization, and Preliminary Antileishmanial Activity. ChemMedChem. 2018, 13(7), 725-735; doi: 10.1002/cmdc.201700770.
- A. Sharma, A. Kumar, S. A. H. Abdel Monaim, Y. E. Jad, Ayman El-Faham, B. G. de la Torre, F. Albericio. N-methylation in amino acids and peptides: Scope and limitations. Biopolymers. 2018; e23110, 1-14; doi.org/10.1002/bip.23110.
- H. H. Al-Rasheed, E. N. Sholkamy, M. Al Alshaikh, M. R. H. Siddiqui , Ahmed S. Al-Obaidi, and Ayman El-Faham. Synthesis, Characterization, and Antimicrobial Studies of Novel Series of 2,4-Bis(hydrazino)-6-substituted-1,3,5-triazine and Their Schiff Base Derivatives. J. Chemistry, Volume 2018, Article ID 8507567, 13 pages, 2018, doi.org/10.1155/2018/8507567.
- D. R. Ramadan, A.A. Elbardan, A.A. Bekhit, Ayman El-Faham, S.N. Khattab. Synthesis and characterization of novel dimeric s-triazine derivatives as potential anti-bacterial agents against MDR clinical isolates. New J. Chem., 2018, 42, 10676-10688; 10.1039/C8NJ01483C.
- M. Farooq, Z. M. Almarhoon, N. Abu Taha, A. A. R. Baabbad, M. A. Al-Wadaan, Ayman El-Faham .Synthesis of novel class of N-alkyl-isatin-3-iminobenzoic acid derivatives and their biological activity in zebrafish embryos and Human cancer cell lines. Biolog. Pharm. Bull.; 2018, 41, 350-359; doi:10.1248/bpb.b17-00674.
- S. A. H. Abdel Monaim, Y. E. Jad, Ayman El-Faham, B. G. de la Torre, F. Albericio. Teixobactin as a scaffold for unlimited new antimicrobial peptides: SAR study. Org. Biomol. Chem., 2018, 16, 5661-5666; doi: 10.1039/C8OB01463A.
- S. M. Soliman and Ayman El-Faham. Low temperature X-ray structure analyses combined with NBO studies of a new heteroleptic octa-coordinated Holmium(III) complex with N,N,N-tridentate hydrazono-phthalazine-type ligand. J. Mol. Str., 2018, 1157, 222- 229. doi.org/10.1016/j.molstruc.
- A. Kumar, Yahya E. Jad, Ayman El-Faham, B. G. de la Torre, F. Albericio. Diethylphosphoryl-OxymaB (DEPO-B) as a Solid Coupling Reagent for Amide Bond Formation. Lett. Org. Chem, 2018, 16 (1), 30-33, doi: 10.2174/1570178615666180612074420.
- S. M. Osman, Sherine N. Khattab, El-Saied A. Aly, El-Refaie Kenawy, Ayman El-Faham. 1,3,5-Triazine-based polymer: synthesis, characterization and application for immobilization of silver nanoparticles. J. Poly. Res., 2017, 24, 231-244; doi.org/10.1007/s10965-017-1385-2.
- S. A. H. Abdel Monaim, S. Noki, E.J. Ramchuran, Ayman El-Faham, F. Albericio and B.G. de la Torre. Investigating of N-terminal amino function of Arg10-teixobactin" Molecules, 2017, 22, 1632; doi:10.3390/molecules22101632
- A. Kumar; A. Sharma; E. Haimov; Ayman El-Faham; B. G. de la Torre; F. Albericio. Fmoc-Amox, A Suitable Reagent for the Introduction of Fmoc. Org. Process Res. Dev. 2017, 21 (10), 1533–154; doi: 10.1021/acs.oprd.7b00199.
- S. M. Soliman, H. A. Ghabbour, S. N. Khattab, M. R. H. Siddiqui, and Ayman El-Faham. Synthesis, crystallographic characterization, DFT and TD-DFT studies of Oxyma-sulfonate esters. J. Chem. Sci., 2017, 129 (9), 1469–1481, doi: 10.1007/s12039-017-1354-7.
- S. A. H. Abdel Monaim, Estelle J. Ramchuran, Ayman El-Faham, Fernando Albericio, and Beatriz G. de la Torre. Converting Teixobactin into a Cationic Antimicrobial Peptide (AMP). J. Med. Chem., 2017, 60(17), 7476-7482, doi: 10.1021/acs.jmedchem.7b00834.
- F. Albericio, G. A. Acosta, Ayman El-Faham, Y. E. Jad, A. Kumar, B. G. de la Torre. Green Solid-Phase Peptide Synthesis (GSPPS). Chimia, 71, No. 7/8 523 (2017).
- A. Kumar, Y. E. Jad, Ayman El-Faham, B. G. de la Torre, F.Albericio. Green Solid-Phase Peptide Synthesis 4. δ-Valerolactone and N-Formylmorpholine as Green Solvents for Solid Phase Peptide Synthesis. Tetrahedron Lett., 2017, 58(30), 2986-2988; doi: 10.1016/j.tetlet.2017.06.058.
- S. M. Soliman, Ayman El-Faham, J. H. Albering. Synthesis, X-ray crystal structure and DFT studies of two octahedral cobalt(II) complexes with N,N,N-tridentate triazine-type ligands. J. Coord.Chem., 2017, 70(13), 2261-2279; doi: 10.1080/00958972.2017.1340646.
- A. Kumar, Y. E. Jad, B. G. de la Torre, Ayman El-Faham, F. Albericio. Re-evaluating the stability of COMU in different solvents. J. Pept. Sci., 2017, 23(10), 763-768; doi: 10.1002/psc.3024.
- A. Sharma, Y. Jad, M. R. H. Siddiqui, B. G. de la Torre, F. Albericio, Ayman El-Faham. Synthesis, Characterization, and Tautomerism of 1,3-Dimethyl Pyrimidine-2,4,6-Trione s-Triazinyl Hydrazine/Hydrazone Derivatives. J. Chem, Volume 2017, Article ID 5702962, 2017, 1-10; doi.org/10.1155/2017/5702962.
- A. Sharma, H. Ghabbour, S.T. Khan, B. G. de la Torre, F. Albericio, Ayman El-Faham. Novel Pyrazolyl-s-Triazine Derivatives, Molecular 1 Structure and Antimicrobial Activity. J. Mol. Str., 2017, 1145, 244-253; doi: 10.1016/j.molstruc.2017.05.040.
- S. M. Soliman and Ayman El-Faham. Synthesis, Crystal Structure and Hirshfeld Topology Analysis of Polymeric Silver(I) Complex with s-Triazine-Type Ligand. Crystals, 2017, 7,160, 1-12, ,; doi:10.3390/cryst7060160.
- S. M. Soliman, J. H. Albering, M. Farooq, M. A. M. Wadaan, Ayman El-Faham. Synthesis, structural and biological studies of two new Co(III) complexes with tridentate hydrazone ligand derived from the antihypertensive drug hydralazine” Inorganica Chimica Acta, 2017, 466, 16–29; doi.org/10.1016/j.ica.2017.05.045.
- Kh. M. Al-Zaydi, H. H. Khalil, Ayman El-Faham, Sh. N. Khattab. Synthesis, characterization and evaluation of 1,3,5-triazine aminobenzoic acid derivatives for their antimicrobial activity. Chem. Cent. J. 2017, 11:39, 1-12; doi:10.1186/s13065-017-0267-3.
- A. Sharma, I. R.-Tomillero, Ayman El-Faham, E. Nicolas, H. Rodriguez, B. G. de la Torre, F. Albericio. Understanding 'Thp' as protecting group in peptide chemistry. ChemistryOpen, 2017, 6, 168 – 177,; doi: 10.1002/open.201600156.
- A. Sharma, I. R.-Tomillero, Ayman El-Faham, H. Rodriguez, B. G. de la Torre., F. Albericio. Tetrahydropyranyl: A non-aromatic, mild acid labile protecting group for hydroxyl protection in Solid Phase Peptide Synthesis. ChemistryOpen, 2017, 6, 206 – 210;doi: 10.1002/open.201600157.
- Y. E. Jad, Th. Govender, H. G. Kruger, Ayman El-Faham, B. G. de la Torre, F. Albericio. Green Solid-Phase Peptide Synthesis (GSPPS) 3. Green Solvents for Fmoc Removal in Peptide Chemistry. Org. Process Res. Dev. 2017, 21, 365−369, doi: 10.1021/acs.oprd.6b00439.
- Sh. N. Khattab, N. S. Haiba, A. M. Asal, A. A. Bekhit, A. A. Guemei, A. Amer, Ayman El-Faham. Study of antileishmanial activity of 2-aminobenzoyl amino acid hydrazides and their quinazoline derivatives. Bioorg. Med. Chem. Lett., 2017, 27, 918–921; doi.org/10.1016/j.bmcl.2017.01.003.
- Sh. N. Khattab, M. I. Massoud, A. M. Abd El-Razek, Ayman El-Faham. Physico-chemical and sensory characteristics of steviolbioside synthesized from stevioside and its application in fruit drinks and food. J. Food, Sci. Technol., 2017, 54(1):185–195 (), doi.10.1007/s13197-016-2450-2.
- A. Sharma , Y. E. Jad, H. A. Ghabbour, B. G. de la Torre, H. G. Kruger, F. Albericio, Ayman El-Faham. Synthesis, Crystal Structure and DFT Studies of 1,3-Dimethyl-5-propionylpyrimidine- 2,4,6(1H,3H,5H)-trione. Crystals, 2017, 7, 31-40 (), doi:10.3390/cryst7010031.
- Ayman El-Faham, Sh. N. Khattab, H. A. Ghabbour. Crystal structure of 1-methyl-3-[((naphthalen-2-ylsulfonyl)oxy)imino]indolin-2-one, C19H14N2O4S. Z. Kristallogr. NCS 2017, 232(1): 55–57. doi: 10.1515/ncrs-2016-0146.
- Ayman El-Faham, A.El-Merghany, H. A. Ghabbour. Crystal structure of N′-(2-phenylacetyl) thiophene-2-carbohydrazide monohydrate, C13H14N2O3S. Z. Kristallogr. NCS, 2017, 232(1): 69–71; doi: 10.1515/ncrs-2016-0152.
- Ayman El-Faham and Hazem A. Ghabbour. Crystal structure of (E)-1-(2-(thiophen-2- ylmethylene)hydrazinyl)phthalazine hydrochloride–ethanol (1/1), C15H17ClN4OS. Z. Kristallogr. NCS, 2017, 232(1): 95–97; doi: 10.1515/ncrs-2016-0168.
- H. H. Al-Rasheed, M. Al Alshaikh, J. M. Khaled, N. S. Alharbi, Ayman El-Faham. Ultrasonic Irradiation: Synthesis, Characterization, and Preliminary Antimicrobial Activity of Novel Series of 4,6-Disubstituted-1,3,5-triazine Containing Hydrazone Derivatives. Journal of Chemistry, Article ID 3464758. Volume 2016, Article ID 3464758, 2016, 1-9; doi.org/10.1155/2016/3464758.
- Sh. A. H. Abdel Monaim, Y.E. Jad, E. J. Ramchuran, Ayman El-Faham, Th. Govender, H.G. Kruger, B. G. de la Torre, and F. Albericio. Lysine Scanning of Arg10−Teixobactin: Deciphering the Role of Hydrophobic and Hydrophilic Residues. ACS Omega, 2016, 1, 1262-1265; doi: 10.1021/acsomega.6b00354.
- Y. E. Jad, G. Acosta, T. Govender, H. Kruger, Ayman El-Faham, B. de la Torre, F. Albericio. Green Solid-Phase Peptide Synthesis-2.1, 2-Methytetrahydrofuran and ethyl acetate for solid-phase peptide synthesis under green conditions.ACS Sustainable Chem. Eng., 2016, 4, 6809−6814; doi: 10.1021/acssuschemeng.6b01765.
- Sh. Khattab, S. E A. Naim, M. El-Sayed, A. A. El Bardan, A. O. Elzoghby, A. A. Bekhit ,Ayman El-Faham. Design and Synthesis of New s-Triazine Polymers and its Application as Nanoparticulate Drug Delivery Systems. New J. Chem., 2016, 40, 9565-9578; doi: 10.1039/C6NJ02539K
- Sh. A. H. Abdel Monaim, Y. E. Jad, G. A. Acosta, T. Naicker, E. J. Ramchuran, Ayman El-Faham,T. Govender, H.G. Kruger, B. G. de la Torre, F. Albericio. Re-evaluation of the N-terminal substitution and the D-residues of teixobactin. RSC Adv., 2016, 6, 73827–73829; doi: 10.1039/c6ra17720d.
- Y. E. Jad, B. G. de la Torre, T. Govender, H.G. Kruger, Ayman El-Faham, F. Albericio. Oxyma-T, expanding the arsenal of coupling reagents. Tetrahedron Letters, 2016, 57, 3523–3525; doi:10.1016/j.tetlet.2016.06.109.
- Ayman El-Faham, S. M. Soliman, H. A. Ghabbour, Y. A. Elnakady, T. A. Mohaya, M. R.H. Siddiqui, F. Albericio. Ultrasonic promoted synthesis of novel s-triazine-Schiff base derivatives; molecular structure, spectroscopic studies and their preliminary anti-proliferative activities. J. Mol. Str., 2016, 1125, 121-135; doi:10.1016/j.molstruc.2016.06.061.
- G. A. El-Mahdy, H. H. Al-Rasheed, M. Al Alshaikh, H. A. Al-Lohedan, Ayman El-Faham. 2,4-Dihydrazino-6-Morpholino-1,3,5-Triaizne (DHMT) and 2,4-Dihydrazino-6-Piperidino-1,3,5-Triaizne (DHPT) as Promising Corrosion Inhibitors of Steel in Acidic Media. Int. J. Electrochem. Sci., 2016, 11, 5459 – 5472; doi: 10.20964/2016.07.08.
- Ayman El-Faham, Kh. A. Dahlous, Z. A. AL Othman, H. A. Al-Lohedan, G. A. El-Mahdy. sym-Trisubstituted 1,3,5-Triazine Derivatives as Promising Organic Corrosion Inhibitors for Steel in Acidic Solution. Molecules, 2016, 21, 436-447; doi:10.3390/molecules21040436.
- Ayman El-Faham, S. M. Osman, H. A. Al-Lohedan, G. A. El-Mahdy. Hydrazino-methoxy-1,3,5-triazine Derivatives Excellent Corrosion Organic Inhibitors of Steel in Acidic Chloride Solution. Molecules, 2016, 21, 714-727; doi:10.3390/molecules21060714.
- M. M.G. Fouda, A. M. Abdel-Mohsen, H. Ebaid, I. Hassan, J. Al-Tamimi, R. M. Abdel-Rahman, A. Metwalli, I. Alhazza, A. Rady, Ayman El-Faham, J. Jancar. Wound healing of different molecular weight of hyaluronan; in-vivo study. Int. J. Biological Macromol. 2016, 89, 582–591; doi: 10.1016/j.ijbiomac.2016.05.021.
- A. M. A. Mashaly and Ayman El-Faham. Larvicidal activity of N1,N1,N4,N4-tetramethylpiperazine-1,4-dicarboxamide against Aedes caspius and Culex pipiens (Diptera: Culicidae). Pakistan J. Zool., 2016, 48 (2), 493-499.
- H. A. Ghabbour and Ayman El-Faham. Crystal structure of 4-chloro-N,N-diethyl-6- (piperidin-1-yl)-1,3,5-triazin-2-amine, C12H20ClN5. Z. Kristallogr. NCS, 2016, 231: 243–245; doi: 10.1515/ncrs-2015-0106
- Ayman El-Faham , S. M. Soliman, S. M. Osman, H. A. Ghabbour, M. R.H. Siddiqui, H.-Kun Fun, F. Albericio. One pot synthesis, molecular structure and spectroscopic studies (X-ray, IR, NMR, UV–Vis) of novel 2-(4,6-dimethoxy-1,3,5-triazin-2-yl) amino acid ester derivatives. Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy, 2016, 159, 184–198; doi.org/10.1016/j.saa.2016.01.051.
- Y. E. Jad · G. A. Acosta, Sh. N. Khattab, B. G. de la Torre1, Th. Govender, H. G. Kruger, Ayman El-Faham, F. Albericio. 2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis. Amino Acids, 2016, 48, 419–426; 10.1007/s00726-015-2095-x.
- Y. E. Jad, G. A. Acosta, T. Naicker, M.Ramtahal, Ayman El-Faham, Th. Govender, H. G. Kruger, B. G. de la Torre, and Fernando Albericio. Synthesis and Biological Evaluation of a Teixobactin Analogue. Org. Lett., 2015, 17, 6182−6185; doi: 10.1021/acs.orglett.5b03176
- S. M. Soliman, M. A. M. Abu-Youssef, J. Albering, Ayman El-Faham. Molecular structure and DFT investigations on new cobalt(II) chloride complex with superbase guanidine type ligand. J. Chem. Sci., 2015, 127 (12), 2137–2149; doi: 10.1007/s12039-015-0976-x.
- Sh. N. Khattab, H. H. Khalil, A. A. Bekhit, M. M. Abd El-Rahman, Ayman El-Faham, F. Albericio. Synthesis and preliminary biological evaluation of 1,3,5-triazine amino acid derivatives to study their MAO inhibitors. Molecules, 2015, 20, 15976-15988; doi:10.3390/molecules200915976.
- Ayman El-Faham, Yasser A. Elnakady. Synthesis, Characterization of Novel Morpholino-1,3,5-triazinyl Amino Acid Ester Derivatives and their Anti-Proliferation Activities. Lett. Org. Chem., 2015, 12, 753-758; doi: 10.2174/1570178612666150709165843
- Ayman El-Faham, W. N. Hozzein, M. A.M.Wadaan, Sh. N. Khattab, H. A. Ghabbour, H.-K. Fun, M. R.Siddiqui. Microwave Synthesis, Characterization, and Antimicrobial Activity of Some Novel Isatin Derivatives. J. Chemistry, Article ID 716987, 2015, Vol.2015, 1- 8; doi: 10.1155/2015/716987.
- M. S. Masoud, Ayman El Faham, H. H. Hamoud, A. E. Alic, H. Beidsas. Spectral studies and solvatochromic behaviour of 1-hydroxy-benzotriazole and 7-Aza-l-hydroxybenzotriazole in presence of different solvents. J. Chem. Pharm. Res., 2015, 7(4), 781-791.
- M. H. El-Newehy, S. M. Osman, M. S. Refat, S.S. Al-Deyab, Ayman El-Faham. Microwave synthesis of copolymers based on itaconic acid moiety and their utility for scavenging of copper (II) and Lead (II). J. Macromol. Sci., Part A: Pure and Applied Chemistry, 2015, 52, 561–576; doi: 10.1080/10601325.2015.1039335.
- Ayman El-Faham, M. Farooq, Sh. N. Khattab, N. Abutaha, M. A. Wadaan, H. A. Ghabbour, H.-K. Fun. Synthesis, Characterization, and Anti-Cancer Activity of Some New N′-(2-Oxoindolin-3-ylidene)-2-propylpentane hydrazide-hydrazones Derivatives. Molecules, 2015, 20, 14638-14655; doi:10.3390/molecules200814638.
- Sh. N. Khattab, N. S. Haiba, A.M. Asal, A. A. Bekhit, A. Amer, H. M. Abdel-Rahman, Ayman El-Faham" Synthesis and Evaluation of Quinazoline Amino Acid Derivatives as Mono Amine Oxidase (MAO) Inhibitors. Bioorg. Med.Chem., 2015, 23, 3574–3585; doi: 10.1016/j.bmc.2015.04.021
- Y. E. Jad, G. Acosta, Sh. Khattab, B. G. De la Torre, T. Govender, G. Kruger , Ayman El-Faham, and F. Albericio. EDC.HCl and Potassium Salts of Oxyma and Oxyma-B as Superior Coupling Cocktails for Peptide Synthesis. Eur. J. Org. Chem., 2015, 3116–3120; doi.org/10.1002/ejoc.201500142.
- Sh. Khattab , Ayman El-Faham, and F. Albericio. Peptide Coupling Reactions. Molecular Pharmaceutics & Organic Process Research, 1-3 (2015).
- Sh.N. Khattab, Sh. A. H. Moneim, A. A. Bekhit , A. El Massry, S. Y. Hassan, Ayman El-Faham, H. E. A. Ahmed, A. Amer. Exploring new selective 3-benzylquinoxaline-based MAO-A inhibitors: Design, synthesis, biological evaluation and docking studies. Eur. J. Med. Chem., 2015, 93, 308-320; doi: 10.1016/j.ejmech.2015.02.020.
- Y. E. Jad, G. Acosta, Sh. Khattab, B. G. De la Torre, T. Govender, G. Kruger , Ayman El-Faham, and F. Albericio. Peptide Synthesis Beyond DMF: THF and ACN as Excellent and Friendlier Alternatives. Org. Biomol. Chem., 2015, 13, 2393-2398, DOI: 10.1039/c4ob02046d.
- Ayman El-Faham , Z. Al Marhoon, A.Abdel-Megeed, Sh.N. Khattab, A. Bekhit, F. Albericio " α-Ketoamino acid ester derivatives as promising MAO inhibitors" Bioorg. Med.Chem.Lett., 2015, 25, 70–74, doi: 10.1016/j.bmcl.2014.11.007.
- M. I. Massoud, Sh. N. Khattab, Y. E. Jad, A. A. Bekhit, Ayman El-Faham. Production and Physico-chemical 1 assessment of new stevia amino acid sweeteners from the natural stevioside. Food Chemistry, 2015, 173, 979-985; doi: 10. 1016/j. Food.chem.2014.10.093.
- Y. E. Jad, Sh. N. Khattab, B. G. de la Torre, Th. Govender, H. G. Kruger, Ayman El-Faham and F. Albericio. TOMBU and COMBU as novel uronium-type peptide coupling reagents derived from Oxyma-B. Molecules, 2014, 19, 18953-18965; doi:10.3390/molecules191118953.
- M. F. Ibrahim, A. A. AL-Karewi, Sh. N. Khattab, E. A. Hamed and Ayman El-Faham. Aminolysis of Isatin and N-Acyl Isatin in Acetonitrile and Mixed Acetonitrile-Water Solvents. Asian J. Chem., 2014, 26, 8029-8038; doi: 10.14233/ajchem.2014.16968
- Z. AL Marhoon, A. Abdel-Megeed , E. N. Sholkamy, M. R. H. Siddiqui and Ayman El-Faham . Synthesis of Phenylcarbamic Acid and 2-(2-Oxo-3-(4-substituted phenylimino)indolin-1-yl) Acetohydrazide Derivatives as a Promising Antifungal Agents. Asian. J. Chem., 2014, 26 (22), 7665-7672; doi.org/10.14233/ajchem.2014.17566.
- Y. E. Jad, Sh. N. Khattab, B. G. de la Torre,T. Govender,H. G. Kruger,Ayman El-Faham and F. Albericio. Oxyma-B, an Excellent Racemization Suppressor for Peptide Synthesis. Org. Biomol. Chem., 2014, 12, 8379-8385; DOI: 10.1039/c4ob01612b.
- M. Farooq, Ayman El-Faham, Sh. N. Khattab, A. M. Elkayal, M. F. Ibrahim, N. Abutaha, A. Baabbad , M. A. M. Wadaan, E. A. Hamed. Biological screening of novel derivatives of valproic acid for anticancer and antiangiogenic properties. Asian Pacific Journal of Cancer Prevention, 2014, 15 (18), 7785-7792, doi:10.7314/APJCP.2014.15.18.7785
- Ayman El-Faham, Sh. N. Khattab, H. A. Ghabbour, H-K Fun and M. R. H.Siddiqui. Microwave irradiation: synthesis and characterization of α-ketoamide and bis (α-ketoamide) derivatives via the ring opening of N-acetylisatin. Chem. Cent. J., 2014, 8:27, 1,10; doi:10.1186/1752-153X-8-27.
- Ayman El-Faham, M. Farooq, Sh. N. Khattab, A. M. Elkayal, M. F. Ibrahim, N. Abutaha, M. Ahmad Wadaan, and E. A. Hamed. Synthesis and Biological Activity of Schiff Base Series of Valproyl, N-Valproyl Glycinyl, and N-Valproyl-4-aminobenzoyl Hydrazide Derivatives. Chem. Pharm. Bull., 2014, 62(6) 591–599; doi: 10.1248/cpb.c14-00143.
- Ayman El-Faham, Y. A. Elnakdy, S. A. M. El Gazzar, M. M. Abd El-Rahman, Sh. N. Khattab. Synthesis, characterization and anti-proliferation activities of novel oximino sulfonate esters. Chem. Pharm. Bull., 2014, 62(4) 373–378; doi: 10.1248/cpb.c13-01005.
- Ayman El-Faham, A. A. Elzatahry, Z. A. AlOthman, E. A. Elsayed. Facile method for the synthesis of silver nanoparticles using 3-hydrazino-isatin derivatives in aqueous methanol and their antibacterial activity. Int. J. nanomedicine, 2014, 4,1167-1174; doi: 10.2147/IJN.S58571
- T. S. AL Gerni, A. M. Ismail, M. AL-Zaben and Ayman EL-Faham. Solvent Effects on the Kinetic and Mechanism of N-Mannich Bases of 3-Hydrazonoindole-2-one. Asian J. Chem., 2014, 26(1) 48-52; doi: 0.14233/ajchem.2014.15316
- Ayman El-Faham, Sh. N. Khattab, R. Subirós-Funosasand F. Albericio. BOP-Ox, BOP-OBt, and BOP-OAt: Novel Organophosphinic Coupling Reagents Useful for Solution and Solid-Phase Peptide Synthesis. J. Pept. Sci., 2014, 20: 1–6; doi: 10.1002/psc.2579.
- Ayman El-Faham, Z. Almarhoon, A. Abdel-Megeed and F. Albericio. Oxyma Pure/DIC: An Efficient Reagent for the Synthesis of a Novel Series of 4-[2-(2-Acetylaminophenyl)-2-oxo-acetylamino] Benzoyl Amino Acid Ester Derivatives. Molecules, 2013, 18, 14747-14759; doi:10.3390/molecules181214747
- Ayman El-Faham, Z. Al Marhoon, A. Abdel-Megeed, M. Siddiqui . An efficient and mild method for the synthesis and hydrazinolysis of N -glyoxylamino acid ester derivatives. J. Chemistry, 2013, Article ID 901745, 2013, 6 pages; doi: 10.1155/2013/901745.
- R.Subirós-Funosas, Ayman El-Faham, and F. Albericio. Low-epimerization Peptide Bond Formation with Oxyma Pure: Preparation of Z-L-Phg-Val-OMe. Org. Synth. 2013, 90, 306-315.
- P. Cherkupally, G. A. Acosta, L. Nieto-Rodriguez, J. Spengler,H. Rodriguez, Sh.N. Khattab, Ayman El-Faham, M. Shamis, Y. Luxembourg, R. Prohens, R.Subiros-Funosas, and F. Albericio. K-Oxyma: a strong acylation-promoting, 2-CTC resin-friendly coupling additive. Eur. J. Org. Chem., 2013, 6372–6378; doi: 10.1002/ejoc.201300777.
- M. Ghazzali, Sh. A.N. Khattab, Y. A. Elnakady, F.A. Al-Mekhlafi, Kh. Al-Farhan, Ayman El-Faham . Synthesis, structure, theoretical calculations and biological activity of sulfonate active ester new derivatives. J. Mol. Str., 2013, 1046, 147-152; doi: 10.1016/j.molstruc.2013.04.025.
- R. Subirós-Funosas, Sh. N. Khattab, L. Nieto-Rodriguez, Ayman El-Faham, F. Albericio. Advances in Acylation Methodologies Enhanced by Oxyma-Based Reagents" Aldrichimica Acta, , 2013, 40 (1), 21-40.
- Ayman El-Faham, Hammed H.A.M. Hassan, Sherine N. Khattab. Synthesis and characterization of new polyamides derived from alanine and valine derivatives. Chem. Cent. J., 2012, 6:128, 1-10; doi:10.1186/1752-153X-6-128.
- S. M. Osman, M. H. El-Newehy, S. S. Al-Deyab, Ayman El-Faham. Microwave synthesis and thermal properties of polyacrylate derivatives containing itaconic anhydride moieties. Chem. Cent. J, 2012, 6:85, 1-10; doi:10.1186/1752-153X-6-85.
- Y. E. Jad, Sh. N. Khattab, Ayman El-Faham, and F. Albericio. Oxime-Based Carbonates as Useful Reagents for Both N-Protection and Peptide Coupling. Molecules, 2012, 17, 14361-14376; doi:10.3390/molecules171214361.
- M. Farooq; Ayman. El-Faham; M. Ahmad, A.S. Sami and M.A. Wadaan. The teratogenic profile of valproic acid (VPA) and newly synthesized derivatives in zebrafish embryos. Int. J. Agric. Biol., 2012, 14: 894‒900; ISSN Print: 1560–8530; ISSN Online: 1814–9596
- Sh. N. Khattab, M. A. H. Kharaba, A. El-Hawary, Ayman El-Faham, E. A. Hamed. Aminolysis of 1-(1-hydroxybenzotriazolyl)-2,4-dinitrobenzene and 2-(1-hydroxybenzotriazolyl)-5-nitro-pyridine. Open J. Phy.Chem. (OJPC), 2012, 2, 156-168; DOI: 10.4236/ojpc.2012.23021
- Sh. N. Khattab, R. Subirós-Funosas, Ayman El-Faham, and F. Albericio. Screening of N-alkyl-cyanoacetamido oximes as Substitutes for N-Hydroxysuccinimide. ChemistryOpen 2012, 1, 147 – 152; doi: 10.1002/open.201200012 .
- H. M. Al-Hazimi, Ayman El-Faham, M. Gazzali, K. Al-Farhan. Microwave irradiation: A facile, scalable and convenient method for synthesis of N-phthaloylamino acids. Arab. J. Chem., 2012, 5, 285-289; doi: 10.1016/j.arabjc.2010.06.020
- Tarfah I. Al-Warhi, Hassan M.A. AL-Hazimi, Ayman El-Faham. Recent Development in Peptide Coupling Reagents. J. S. Chem. Soc., 2012, 16, 97-116; doi: 10.1016/j.jscs.2010.12.006
- Sh. N. Khattab, R. Subirós-Funosas, Ayman El-Faham, F. Albericio. Cyanoacetamide-based oxime carbonates: an efficient, simple alternative for the introduction of Fmoc with minimal dipeptide formation. Tetrahedron, 2012, 68, 3056-3062; doi:10.1016/j.tet.2012.02.020.
- M. Ghazzal, Ayman El-Faham, A. Abd-Megeed, Kh. Al-Farhan. Microwave-assisted synthesis, structural elucidation and biological assessment of 2-(2-acetamidophenyl)-2-oxo-N phenyl acetamide and N-(2-(2-oxo-2(phenylamino)acetyl)phenyl)propionamide derivatives. J. Mol. Str., 2012, 1013, 163-167; doi:10.1016/j.molstruc.2012.01.028.
- R. Subiros-Funosas, Ayman El-Faham, F. Albericio. Use of Oxyma as pH modulatory agent to be used in the prevention of base-driven side reactions and its effect on 2-chlorotrityl chloride resin. Biopolymer (Peptide Science) 2012, 98 (2), 89-97; doi: 10.1002/bip.21713
- H. H. A. M. Hassan, A. F. El-Husseiny, A. G. Abo ElFadl, Ayman El-Faham, and F. Albericio .Synthesis and Thermal Properties of Novel Polyamides Containing Amino Acid Moities: Structure-Property Relationship. J. Macromol. Sci., Part A: Pure and Applied Chemistry, 2012, 49, 41–54, doi: 10.1080/10601325.2012.630935
- Ayman El-Faham and Fernando Albericio. Peptide Coupling Reagents, More than a Letter Soup. Chem. Rev., 2011, 111, 6557–6602; doi: 10.1021/cr100048w
- R. Subiros-Funosas, Ayman El-Faham, F. Albericio. Aspartimide formation in peptide chemistry: occurrence, prevention strategies and the role of N-hydroxylamines. Tetrahedron, 2011, 67, 8595-8606; doi:10.1016/j.tet.2011.08.046.
- Sh. N. Khattab, E. A. Hamed, F. Albericio, and Ayman El-Faham. Synthesis and aminolysis of N, N, Diethyl Carbamic ester of HOBt. Bull. Chem. Soc., Jpn. 2011, 84, 633-639; doi:10.1246/bcsj.20110015.
- Kh. Al-Farhan, M. Ghazzali, H. M.A. Al-Hazimi, Ayman El-Faham, J. Reedijk. Hydrogen bonding chains and rings structural motifs in new series of N-phthaloyl aminocarboxylic acid derivatives. Solid state microwave synthesis, structural chemistry, computational calculations and antimicrobial activity. J. Mol. Str., 2011, 994, 269–275; doi:10.1016/j.molstruc.2011.03.030.
- Tarfah I. Al-Warhi, Hassan M.A. AL-Hazimi, Ayman El-Faham and Fernando Albericio. Synthesis of 2-(4,6-Dimethoxy-1,3,5-triazin-2-yloxyimino) Derivatives: Application in Solution Peptide Synthesis. Molecules, 2010, 15, 9403-9417; doi:10.3390/molecules15129403.
- M. Albatal, M. Abdul Ghani, Ayman El-Faham, H. M. Al-Hazimi, H. H. Hammud. Microwave Irradiation and Diisopropylcarbodiimide (DIC)/7-Aza-1- hydroxyl benzotriazole (HOAt): A Potent Combination for Synthesis of Various Hydrazide from N-Protected Amino Acid and Hydrazine. J. Korean. Chem. Soc., 2010, 54, 419-428.
- M. Ghazzali, K. Al-Farhan, Ayman El-Faham, J. Reedijk. Coordination chemistry of the ligand 7-aza-1-hydroxy-benzotriazole. Crystal structures and antimicrobial activity of the catena-poly-[μ-chlorido(μ-7-aza-1-oxy-κ2N:O-benzotriazolyl-κN)]cobalt(II)methanol coordination polymer and of a new polymorph of the free ligand 3H-[1,2,3]triazolo[4,5-b]pyridin-3-ol. Polyhedron, 2010, 29, 2829–2832; doi:10.1016/j.poly.2010.07.004.
- R. Subiros-Funosas, Ayman El-Faham, F. Albericio. PyOxP and PyOxB: the Oxyma-based novel family of phosphonium salts. Org. Biomol. Chem., 2010, 8, 3665–3673; doi: 10.1039/c003719b.
- Ayman El-Faham, R. Subiros-Funosas and F. Albericio. A novel family of onium salts based upon isonitroso Meldrum´s acid proves useful as peptide coupling reagents. Eur. J. Org. Chem. 2010, 3641-3649; DOI: 10.1002/ejoc.201000314.
- Sh. N. Khattab, R. Subirós-Funosas, Ayman El-Faham, F. Albericio. Oxime Carbonates, Novel Reagents for the Introduction of Fmoc and Alloc Protecting Groups, Free of Side-Reactions. Eur. J. Org. Chem., 2010, 3275–3280; doi: 10.1002/ejoc.201000028
- Ayman El-Faham and Fernando Albericio. COMU:” A Third Generation of Uronium-Type Based Coupling Reagent. J. Peptide Sci. 2010, 16, 6-9; doi: 10.1002/psc.1204.
- Sh. N. Khattab, S.Y. Hassan, E. A. Hamed, F. Albericio and Ayman El-Faham. Synthesis and aminolysis of N, N, Diethyl Carbamic ester of HOBt. Bull. Korean Chem. Soc., 2010, 31, 75-81; doi: 10.5012/bkcs.2010.31.01.075
- R. Subiros-Funosas, G. A. Acosta, Ayman El-Faham, F. Albericio. Microwave irradiation and COMU: a Superior tool for solid phase peptide synthesis" Tetrahedron Lett. 2009, 50, 6200-6202; doi:10.1016/j.tetlet.2009.08.117.
- L. A. Carpino, K. Nasr, A. A. Abdel-Maksoud, Ayman El-Faham, D. Ionescu, O P. Henklein, H. Wenschuh, M. Beyermann, E. Krause, and M. Bienert. Dicyclopropylmethyl Peptide Backbone Protectant. Org. Lett., 2009, 11, 3718-3721; doi: 10.1021/ol901310q.
- R. Subirós-Funosas, R. Prohens, R. Barbas, Ayman El-Faham, F. Albericio. Oxyma: an efficient additive for peptide synthesis to replace benzotriazole-based HOBt and HOAt with a lower risk of explosion. Chem. Eur. J., 2009, 15, 9394 – 9403; doi: 10.1002/chem.200900614.
- Ayman El-Faham, R. Subirós-Funosas, R. Prohens, F. Albericio. COMU, a Safer and More Effective Replacement for Benzotriazole-based Uronium Coupling Reagents. Chem. Eur. J., 2009, 15, 9404 – 9416; doi: 10.1002/chem.200900615.
- H. H. Hammud, K. T. Holman, M. S. Masoud, Ayman El-Faham, H. Beidas. 1-Hydroxybenzotriazole (HOBt) acidity, formation constant with different metals and thermodtnamic parameters. Synthesis and characterization of Some HOBt metal complexes. Crystal structures of two polymers:[Cu2(H2O)5(HOBt)2(µ -OBt)2].2H2O.EtOH(1A) and [Cu(µ-OBt)(HOBt)(OBt)(EtOH](1B). Inorganic Chimica Acta, 2009, 362, 3526-3540; doi:10.1016/j.ica.2009.03.046.
- Ayman El-Faham and Sh. N. Khattab. Utilizations of Fluoroformamidinium Salts in Peptide and Organic Syntheses. Synlett., 2009, 886-904; doi:10.1016/j.ica.2009.03.046
- Ayman El-Faham and Fernando Albericio. Synthesis and Application of N-hydroxyamine Derivatives as Potential Replacement for HOBt. Eu. J. Org. Chem. 2009, 1499-1501; doi: 10.1002/ejoc.200801179.
- Ayman El-Faham and Fernando Albericio. Morpholine-Based Immonium and Halogenoamidinium Salts as Coupling Reagents in Peptide Synthesis. J. Org. Chem, 2008, 73, 2731-2737; doi: 10.1021/jo702622c.
- Ayman El-Faham, Mercedes Armond Ugon, Jose A. Este and Fernando Albericio. Use of N-Methyl piperazine for the Preparation of Piperazino-Based Unsymmetrical Bis-Ureas as Anti-HIV Agents. ChemMedChem., 2008, 3, 1-4; doi: 10.1002/cmdc.200800059
- Sh. N. Khattab, S. Y. Hassan, A. A. Bekhit, A. Amer, Ayman El-Faham. Synthesis of Some Pyridazineacetic Acid Derivatives as a Novel Class of Mono Oxidase-A Inhibitors.Chem. Pharm. Bull. 2008, 56 (12) 1717-1721; doi: 10.1248/cpb.56.1717.
- Sh. Khattab, S. Y. Hassan, Ayman El-Faham, Abdel Moneim M. El-Massry and A. Amer. The Reaction of Phthaladehydic Acid with Different substituted Aniline as well as Hydrazine Derivatives. J. Heterocycl. Chem., 44, 617-626 (2007).
- S. Y. Hassan, Sh. N. Khattab, E. A. Hamed and Ayman El-Faham. Synthesis and aminolysis of N,N-diethylcarbamate ester derivatives of HOAt, HOBt, and 4-HOAt. J. Chem. Research , April, 247-251 (2007).
- S. Y. Hassan, Sh. N. Khattab, and Ayman El-Faham. microwave Synthesis of some 1,2,4-Triazole Derivatives. Bull. Fac. Sci. Alex. Uni., 45, 49-60 (2007).
- Ayman El-Faham and Fernando Albericio. Novel Proton Acceptor Immonium-Type Coupling Reagents: Application in Solution and Solid Phase Peptide Synthesis. Org. Lett., 9, 4475-4477 (2007).
- Ayman El-Faham, Sherine N. Khattab, and Mohamed Abdul-Ghani .Tetramethylfluoro formamidinium hexafluorophosphate (TFFH)/ benzyltriphenyl phosphonium dihydrogen trifluride (PTF) a unique reagent for the conversion of carboxylic acids to the corresponding alcohols as well as hydroxamic acids. Arkivoc, xiii, 57-63 (2006).
- Ayman El-Faham, Sh. N. Khattab, M. Abdul-Ghani, and Fernando Albericio. Design and Synthesis of New Immonium-Type Coupling Reagents” Eu. J. Org. Chem., 6, 1563-1573 (2006).
- Ayman El-Faham, M. R. Chebbo, M Abdul Gahni, and G. O. Younse . Chloroformamidinium Salts: Efficient Reagents for Preparation of 2-Aminobenzoimidazole, 2-Aminobenzoxazole, and 2-Aminobenzothiazole Derivatives. J. Heterocycl. Chem., 43, 1-8 (2006).
- L. A. Carpino, J. Xia, C. Zhang and Ayman El-Faham. Organophoshorus and Nitro- substituted Sulfone Esters of 1-Hydroxy-7-azabenzotriazole as Highly Efficient Fast-Acting Peptide Coupling Reagents. J. Org. Chem., 69, 69-71 (2004).
- L. A. Carpino, J. Xia, and Ayman El-Faham “3-Hydroxy-4-oxo-3, 4-dihydro-5-azabenzo-1,2,3-triazene. J. Org. Chem., 69, 54-61 (2004).
- M. Abdul-Ghani, Sh. N. Khattab, A. M. El Massry, Ayman. El-Faham, and Adel Amer. A Novel and Direct Method for Preparation of 4-Amino-1,1,3,3-TetraSubstituted Guanidines as well as [1,2,4] Triazolo Fused Heterocyclic Derivatives. Org. Prep.Perocd. Int., 36, 121-127 (2004).
- Sh. N. Khattab, A. M. M. El Massry, Ayman El-Faham, A. A. Bekhit and A. Amer. Coupling Reactions of Hydralazine with Amino Acids and their Adducts for Antihypertensive Activities. J. Heterocycl. Chem., 41, 387-392 (2004).
- Ayman El-Faham and M. Abdul Ghani. TFFH: A Convenient Activator for Converting Carboxylic Acids into Acid Amides, Hydrazides, and Azides” Org. Prep. Proced. Int., 35, 369-374 (2003).
- L. A. Carpino, D. Ionescu, Ayman El-Faham, M. Beyerman, P. Henklein, C. Hanay, H. Wenschuh, M. Bienert. Complex Polyfluoride Additive in Fmoc-Amino Acid Fluoride Coupling Processes. Enhanced Reactivity and Avoidance of Stereomutation. Org. Lett., 7, 975-977 (2003).
- Ayman El-Faham. O-(7-azabenzotriazol-1-yl)-1,3-dimethyl-1,3-dimethylene- uronium Hexafluorophosphate. Contribution for: Electronic Encyclopedia of Reagents for Organic Synthesis. (L.A. Paquette, ed.), John Wiley & Sons Ltd, Chichester, U.K., www.mrw.interscience.wiley.com/eros/. (2002).
- Ayman El-Faham. 1,1,3,3-Tetramethylfluoroformamidinium Hexafluoro- phosphate. Contribution for: Electronic Encyclopedia of Reagents for Organic Synthesis. (L.A. Paquette, ed.), John Wiley & Sons Ltd, Chichester, U.K., www.mrw.interscience.wiley.com/eros/ (2002)
- L. A. Carpino, H. Imazumi, Ayman El-Faham, et al. The Uronium/ Guanidinium Peptide Coupling Reagents: Finally the True Uronium Salts" Angew. Chem. Int. Ed. 41, 441-445 (2002).
- Ayman El-Faham, A. M. El-Massry, A. Amer, Y. Goher. Versatile Synthetic Route to Chiral Quinoxaline from Amino Acids Precursors. Lett. Pept. Sci. 9, 49-54 (2002).
- L. A. Carpino, P. Henklein, B. M. Foxman, I. Abdelmoty, B. Costisella, V. Wray, T. Domke, Ayman El-Faham, and C. Mugge. The Solid and Solution Structure of HAPyU. J. Org. Chem., 66, 5245-5247 (2001).
- Sh. N. Khattab, Ayman El-Faham, A. M. El-Massry, E. M. E. Mansour, M. M. Abd El-Rahman .Coupling of Iminodiacetic Acid with Amino Acid Derivatives in Solution and Solid phase. Lett. Pept. Sci., 7, 331-345 (2001).
- M. del Fersno, Ayman El-Faham, L. A. Carpino, M. Royo and F. Albericio. Substituted Guanidines: Introducing Diversity In Combinatorial Chemistry. Org. Lett., 2, 3539-3542 (2000).
- Ayman El-Faham. Addition of HOXt (X=A or B) Improve the Effeciency of Phenol-Based Coupling Reagents during Peptide Synthesis. Lett. Pept. Sci., 7, 113-121 (2000).
- L. A. Carpino, H. Imazumi, B. M. Foxman, M. J. Vela, P. Henklein, Ayman El-Faham, J. Klose and M. Bienert. Comparison of the Effects of 5- and 6-HOAt on Model Peptide Coupling Reactions Relative to the Cases for the 4- and 7-Isomers. Org. Lett., 2, 2253-2256 (2000).
- L. A. Carpino, M. Ismail, G. A. Truran, E. M. E. Mansour, S. Iguchi, D. Ionscu, Ayman El-Faham, C. Reimer, and R. Warrass. The 1, 1-Dioxobezo[b] thiophene-2-ylmethyloxycarbonyl (Bsmoc) Amino-Protecting Group. J. Org. Chem., 64, 4324-4338 (1999).
- L. A. Carpino and Ayman El-Faham. The Diisopropylcarbodiimide/1-Hydroxy- 7- azabenzotriazole System: Segment Coupling and Stepwise Peptide Assembly. Tetrahedron, 55, 6813-6830 (1999).
- J. Klose, Ayman El-Faham, P. Henklein, L. A. Carpino, and M. Bienert. Addtion of HOAt Dramatically Improve the Effectiveness of Pentafluorophenyl-Based Coupling Reagents. Tetrahedron. Lett., 40, 2045-2048 (1999).
- L. A. Carpino, D. Ionescu, Ayman El-Faham, P. Henklein, H. Wenschuh, M. Bienert, and M. Beyermann. Protected Amino Acid Chlorides vs Protected Amino Acid Fluorides: Reactivity Comparisons. Tetrahedron Lett., 39, 241-244 (1998).
- Ayman El-Faham. Bis(tetramethylene)fluoroformamidinium Hexafluoro- phosphate (BTFFH): A Convenient Coupling Reagent in Solid Phase Peptide Synthesis. Chemistry Lett., 7, 671-672 (1998).
- Ayman El-Faham. New Syntheses of bis(tetramethylene)fluoroformamidinium Hexafluorophosphate (BTFFH) and 1,3-Dimethyl-2-fluoro-4,5-dihydro-1H-imid- azolium Hexafluorophosphate (DFIH). Utility in Peptide Coupling Reactions. Org. Prep. Procd. Int., 30, 477-481 (1998).
- F. Albericio, J. M. Bofill, Ayman El-Faham, and S. A. Kates. On the Use of Onium Salt-Based Coupling Reagents in Peptide Synthesis. J. Org. Chem., 63, 9678-9683 (1998).
- L. A. Carpino, M. Philbin, M. Ismail, G. A. Truran, E. M. E. Mansour, S. Igushi, D. Ionescu, Ayman El-Faham, C. Riemer, R. Warrass, and M. Weiss. New Family of Bases and Nucleophile-Sensitive Amino-Protecting Groups. A Michael-Acceptor-Based Deblocking Process. Practical Utilization of the 1,1-Dioxobenzo[b]thiophene-2-ylmethyloxycarbonyl (Bsmoc) Group. J. Am. Chem. Soc., 119, 9915-9916 (1997).
- E. A. Hamed, Ayman El-Faham, A. A. El-Bardan, and E. F. Saad. Synthesis and Spectral Studies of Some Aryl Sulfides and Sulfones” Journal of Phosphorus, Sulphur, and Silicon, 119, 11-26 (1996).
- E. F. Saad, E. A. Hamed, and Ayman El-Faham. Spectral Characterization of Some Phenylazodihydroxynaphthalene Derivatives. Spectroscopy Lett., 29, 1047-1065 (1996).
- L. A. Carpino, D. Ionescu, and Ayman El-Faham. Peptide Coupling in the Presence of Highly Hindered Tertiary Amines. J. Org. Chem., 61, 2460-2465 (1996).
- Ayman El-Faham. Azabenzotriazolyluronium Salt as a New Coupling Reagent in Peptide Synthesis. Bull. Fac. Sci. Alex. Univ., 36, 73-80 (1996); Chem. Abs., 125, 11428w (1996).
- L. A. Carpino, H. G. Chao, S. Ghassemi, E. M. E. Mansour, C. Riemer, R. Warrass, D. Sadat-Aalaee, G. A. Truran, H. Imazumi, Ayman El-Faham, D. Ionescu, M. Ismail, T. L. Kowaleski, C. H. Han, H. Wenschuh, M. Beyermann, M. Bienert, H. Shroff, F. Albericio, S. A. Triolo, N. A. Sole, and S. A. Kates. Novel Carboxylic Acid Carboxamide Protective Groups Based on the Exceptional Stabilization of the Cyclopropylmethyl Cation. J. Org. Chem., 60, 7718-7719 (1995).
- L. A. Carpino, Ayman El-Faham, and F. Albericio. Efficiency in Peptide Coupling: 1- Hydroxy-7-azabenzotriazole vs 3, 4-Dihydro-3-hydroxy-4-oxo-1,2,3-benzotriazine” J. Org. Chem., 60, 3561-3564 (1995).
- A. A. Kassem, Ayman El-Faham, and H. A. El-Wakil. Aroylhydrazide and Hydrazone Derivatives of Fluorene-9-yl-derivatives. International J. Chem., 6, 5-10(1995); Chem. Abs., 125, 86281b (1995).
- H. Wenschuh, M. Beyermann, Ayman El-Faham, S. Ghassemi, L. A. Carpino, and M. Bienert “Peptide Assembly in the Absence of Base via FMOC Amino Acid Fluorides. J. Chem. Soc., Chem. Commun., 669-670 (1995).
- L. A. Carpino and Ayman El-Faham. Tetramethylfluoroformamidinium Hexafluoro phosphate: A Rapid-Acting Peptide Coupling Reagent for Solution and Solid Phase Peptide Synthesis. J. Am. Chem. Soc., 117, 5401-5402 (1995).
- H. Wenschuh, M. Beyermann, H. Haber, J. K. Seydel, E. Krause, M. Bienert, L. A. Carpino, Ayman El-Faham, and Fernando Albericio. Stepwise Automated Solid Phase Synthesis of Naturally Occurring Peptaibols Using FMOC Amino Acid Fluorides. J. Org. Chem., 60, 405-410 (1995).
- L. A. Carpino, Ayman EL-Faham, and Fernando Albericio. Racemization Studies During Solid Phase Peptide Synthesis Using Azabenzotriazole-Based Coupling Reagents. Tetrahedron Lett., 35, 2279-2282 (1994).
- L. A. Carpino and Ayman El-Faham. Effect of Tertiary Bases on O-Benzotri- azolyluronium Salt-Induced Peptide Segment Coupling. J. Org. Chem., 59, 695-698 (1994).
- L. A. Carpino, Ayman El-Faham, Charles. A. Minor, Fernando Albericio. Advantageous Applications of Azabenzotriazole (Triazopyridine)-Based Coupling Reagents to Solid Phase Peptide Synthesis. J. Chem. Soc., Chem. Commun., 201-203 (1994).
- L. A. Carpino, E. M. E. Mansour, and Ayman El-Faham. Bis(Boc) Amino Acid Fluorides as Reactive Peptide Coupling Reagents. J. Org. Chem., 58, 4162-4164 (1993).
IV- Conference Publications
- Fernando Albericio, Ayman El-Faham, Beatriz G. de la Torre “Solid-Phase Peptide Synthesis: Being Greener, Being Better” TIDES: Oligonucleotide and Peptide Therapeutics, May 20, 2019; San Diego (CA, USA)
- Ayman El-Faham, Zainab Almarhoon, Beatriz G. de la Torre, and Fernando Albericio " Chemoselectivity of cyanuric chloride (TCT) as a trifunctional linker with different nucleophiles"7th Annual International Conference on Chemistry, 22-25 July 2019, Athens, Greece
- Ayman El-Faham, Zainab Almarhoon, Yahya E. Jad, Ashish Kumar, Gerardo A. Acosta, Beatriz G. de la Torre, and Fernando Albericio " Recent Progress in Peptide Coupling Reagents and Greener Solvents in Peptide Synthesis"6th Annual International Conference on Chemistry, 23-26 July 2018, Athens, Greece.
- B. de la Torres, S.A. Monaim, Y. Jad, E Ramchuran, Ayman El-Faham, F Albericio"Teixobactin: A recently discovered antimicrobial peptide. Structure-activity relationship" Abstracts of Papers, 255th ACS National Meeting & Exposition, New Orleans, LA, United States, March 18-22, 2018 (2018), MEDI-105.
- F. Albericio, S.A. H. Abdel Monaim , Y. E. Jad, G. A. H. Acosta, E. J. Ramchuran, Ayman El-Faham , Th. Govender, H. G. Kruger and B. G. de la Torre " Structure-Activity Relationship of Arg10-Teixobactin: A Recently Discovered Antimicrobial Peptide" Presented at the 1st Molecules Medicinal Chemistry Symposium, Barcelona, Spain, 8 September 2017; Proceedings 2017, 1, 671; doi:10.3390/proceedings1060671.
- S. A. H. Abdel Monaim, Y. E. Jad,1G. A. Acosta,T. Naicker,E. J. Ramchuran, Ayman El-Faham,T. Govender,H. G. Kruger,B. G. de la Torre1and F. Albericio" Structure- Activity Relationship of Arg10-Teixobactin" Frank Warren Conference 2016 Rhodes University –South Africa, P-ABR-790.
- F. Albericio, G. A. Acosta, J. B. Blanco-Canosa,V. Castro, P.Cherkupally, Ayman El- Faham, A.-I.Fernandez-Llamazares, M. Gongora-Benitez, Sh. N. Khattab, T. M. Postma, R.Subiros-Funosas, L. Nieto-Rodriguez, H. Rodriguez, J. Spengler, J.Tulla-Puche" Recent Tricks in Solid-Phase Peptide Synthesis"4th Modern Solid Phase" Peptide Synthesis and its Applications Symposium, Kobe (Japan); 112013. 2015.
- Ayman El-Faham,Y. E. Jad, Sh. N. Khattab, B. G. de la Torre, T. Govender, H. G. Kruger, F. Albericio" OXYMA-B AND ITS URONIUM SALTS: SUPERIOR PEPTIDE COUPLING REAGENTS" BIT's 8th Annual World Protein & Peptide Conference, Nanjing·China, April 25- 28 (2015).
- N. S. Haib, Sh. N. Khattab, A. M. Asal, A. A. Bekhit, A. Amer, Ayman El-Faham" Isatoic anhydride: precurser molecule for preparation of nonpeptide derivatives as MAO- A inhibitors" The 13th IBN SINA International Conference on Pure and Applied Heterocyclic Chemistry, 14 - 17 February, Hurghada, Egypt, 2015.
- H. H. Khalil, Sh. N. Khattab, A. A. Bekhitb, M. M. Abd El- Rahman, Ayman El-Faham, F. Albericio" 1,3,5-Triazinyl amino acid derivatives as potent monoamine oxidase (A and B) inhibitors (MAOI’s A and B)" The 13th IBN SINA International Conference on Pure and Applied Heterocyclic Chemistry, 14 - 17 February, Hurghada, Egypt, 2015.
- Sh. N. Khattab, Ayman El-Faham, Y. Abbas Elnakdy, S. A. M. El Gazzar, M. M. Abd El-Rahman" Synthesis of new cyano oximino sulfonate esters with possible antiproliferation Activities" The 13th IBN SINA International Conference on Pure and Applied Heterocyclic Chemistry, 14 - 17 February, Hurghada, Egypt, 2015.
- Sh. A. H. Abdel Monaim, Sh. N. Khattab, A. A. Bekhit, A. M. El Massry, S. Y. Hassan, Ayman El-Faham, A.Amer" Synthesis of some Quinoxaline Derivatives as Potential Monoamine Oxidase (MAO) Inhibitors" The 13th IBN SINA International Conference on Pure and Applied Heterocyclic Chemistry, 14 - 17 February, Hurghada, Egypt, 2015.
- Y. E. Jad, Sh. N. Khattab, B. G. de la Torre, T. Govender, H. G. Kruger, Ayman El- Faham and F. Albericio "DEVELOPMENT OF NOVELS PEPTIDE COUPLING REAGENTS BASED ON 1,3-DIMETHYLBARBUTRIC ACID, THE OXYMA-B FAMILY" European Peptide symposium 2014
- Y. E. Jad, G. A. Acosta, Sh. N. Khattab, B. G. de la Torre, T. Govender, H. G. Kruger, Ayman El-Faham and F. Albericio "USING ACETONITRILE AND TETRAHYDROFURAN INSTEAD OF N,N-DIMETHYLFORMAMIDE IN PEPTIDE BOND FORMATION" European Peptide symposium 2014
- Ayman El-Faham , Sh. N. Khattab, Ramon Subirós-Funosas, Fernando Albericio " Oxyma Family: Strong, safe, promoting coupling reagents in solution and solid phase peptide synthesis" the 2nd Annual International Conference on Chemistry, Chemical Engineering and Chemical Process (CCECP 2014) to be held on 3rd – 4th February 2014 in Singapore.
- Sh. N. Khattab,] Ramon Subirós-Funosas, Ayman El-Faham Fernando Albericio "mOrganophosphinic Coupling Reagents in Peptide Synthesis " the 2nd Annual International Conference on Chemistry, Chemical Engineering and Chemical Process (CCECP 2014) to be held on 3rd – 4th February 2014 in Singapore.
- L. Nieto-Rodriguez, M. Carceller, R. Subirós-Funosas, G. A. Acosta, M. Paradís Bas, Ayman El-Faham, and F.Albericio ," Practical Tips on the Use of Oxyma: An Exhaustive Stability Assay" Proceedings of the 22nd American Peptide Symposium Michal Lebl (Editor) American Peptide Society, San Diego, CA, U.S.A.2011, pp16-17.
- R. Subirós-Funosas, Ayman El-Faham, and F.Albericio "Novel Applications of Oxyma: Minimization of Base-Driven Side Reactions" Proceedings of the 22nd American Peptide Symposium Michal Lebl (Editor) American Peptide Society, San Diego, CA, U.S.A. 2011, pp18-19.
- F. Albericio, Ayman El-Faham, M. Gongora-Benitez, R. Subirós-Funosas, and J. Tulla-Puche" Solid-Phase Peptide Synthesis: State of the Art" Proceedings of the 22nd American Peptide Symposium Michal Lebl (Editor) American Peptide Society, San Diego, CA, U.S.A. 2011, pp406-407.
- Ayman El-Faham, Ramon Subirós-Funosas, Fernando Albericio “Morpholino Based Coupling Reagent” International meeting for Applied and Pure Chemistry, Sharjah, Emirates, March, 2011.
- Ayman El-Faham, Hassan Al-Hazimi, Ramon Subiros-Funosas, Fernando Albericio “AThird Generation of Uronium and Phosphonium Type-Based Coupling Reagent.” 3rd International PepCon-2010, March 21-23, 2010 in Beijing, China, pp524.
- Ayman El-Faham, Ramon Subirós-Funosas, Fernando Albericio"A Non-Explosive Replacement for Benzotriazole Based Coupling Reagents” in Proceeding of the 30th European Peptide Symposium, 2008.
- Ramon Subirós-Funosas, Ayman El-Faham, , Fernando Albericio" Oxyma Pure :A Potent and Non-Explosive Substituent for the Classical Benzotriazole-based Additives” in proceeding of the 30th European Peptide Symposium, 2008, p57.
- Ayman El-Faham and Fernando Albericio “Proton Acceptor Coupling Reagents: Application in Solution and Solid Phase Peptide Synthesis” Peptide for Youth, " Peptide, Protein, and Peptidomimetic Synthesis, (Eds. Emanuel Escher, William D. Lubell, Susan Del Valle, in Proceeding of the 20th American Peptide Symposium, Canada, 2007, p451
- L. A. Carpino, H. Imazumi, Ayman El-Faham, et al."The Uronium/ Guanidinium Peptide Coupling Reagents: Finally the True Uronium Salts" 18th American Peptide Symposium, Boston, Massachusetts, July 19-23, 2003 pp 349.
- Ayman El-Faham and M. Abdul Ghani” Novel Synthesis and Spectral Characterization of Pentasubstituted Guanidine” International Conference on Research Trends in Science and Technology, March, Beirut, Lebanon, 2002, p49-56.
- Ayman El-Faham and M. Abdul Ghani” TFFH: A Convenient Activator for the Synthesis of Alcohol and N, N’-Diaroylhydrazide” International Conference on Research Trends in Science and Technology, March, Beirut, Lebanon, 2002, p41-47.
- Ayman El-Faham and L. A. Carpino “b-Naphthylsulphonyl Derivatives of HOAt as Coupling reagents in Peptide Synthesis” 7th IBN SINA International Conference on Pure and Applied Heterocyclic Chemistry. (Eds. El-Sayed. H. El-Ashry, A. Kassem, and S. Kholeif) Alexandria, 2000, P 341.
- Sh. Khattab, A. M. El-Massri, Ayman El-Faham “ Synthesis of some Biologically Active Peptides containing Iminodiacetic acid” 7th IBN SINA International Conference on Pure and Applied Heterocyclic Chemistry. (Eds. El-Sayed. H. El-Ashry, A. Kassem, and S. Kholeif) Alexandria, 2000, P 341.
- M. M. Abd El-Rahman, E. M. E. Mansour, A. M. El-Massry, Ayman El-Faham, and Sh. N. Khattab, “Synthesis of Amino Acid Derivatives of Iminodiacetic Acid”, 40th Science Week, proceeding of Basic Sciences, University of Tachreen, 4-9 November 2000, Book 2-part 2, p 525-537
- M. del Fersno, M. Royo, Ayman El-Faham, L. A. Carpino, and F. Albericio "Substituted and non-Substituted Guanidines: Introducing Diversity In Combinatorial Chemistry" in Prceeding of the 26th European Peptide Symposium (Eds. J. Martinz and J. A. Fehrentz ) Editions Medicales et Scientifiques, Paris (France), 2000.
- S. A. Triolo, D. Ionescu, H. Wenschuh, N. A. Sole, Ayman El-Faham, L. A. Carpino, and S. A. Kates “Recent Aspects of the Use of Tetramethylfluoro- formamidinium Hexafluorophosphate (TFFH) as a Convenient Peptide Coupling Reagent” Proceeding of the European Peptide Symposium (Eds. R. Ramage and R. Eplon) Edinburgh, Scotland, The European Peptide Society, 1998, pp 839-840.
- P. Henklein, B. Costisella, V. Wary, T. Domke, L. A. Carpino, Ayman El-Faham, S.Kates, I. Abdelmoty, and B. M. Foxman “ Crystal and Solution Structure of HBPyU and HAPyU” Proceeding of the European Peptide Symposium (Eds. R. Ramage and R. Eplon)The European Peptide Society, 1998, pp 465-466.
- J. Klose, Ayman El-Faham, P. Henklein, L. A. Carpino, and M. Bienert “ Comparison of Various HOAt- and HOPfp-Based Coupling Regaents in Effecting Peptide Cyclization” in Proceeding of the 25th European Peptide Symposium ( Eds S. Bajusz and F. Hudecz) Budapest, 1998, pp 204-205.
- M. Beyermann, D. Ionescu, P. Henklein, Ayman El-Faham, H. Wenschuh, M. Bienert, and L. A. Carpino “ Protected Amino Acid Chlorides: Coupling Reagents Suitable for the most Highly Hindered system” In proceeding the 15th American Peptide Symposium (Eds J.P.Tam and P.T.P. Kaumayal) Nashville, 1997, pp239-240.
- S. A. Kates, S. A. Triolo, G. W. Griffin, L. W. Herman, G. Tarr, N. A. Sole, E. Diekmann, Ayman El-Faham, D. Ionescu, F. Albericio, and L. A. Carpino, “Advances in The Use of Onium-Based Coupling Reagents: Application for Solid Phase Peptide Synthesis and Combinatorial Libraries” in Fourth International Symposium on Solid Phase Synthesis & Combinational Libraries” (Ed. R. Epton) Mayflower Worldwide Scientific Ltd., Birmingham, 1996, pp 41-50.
- E. A. Hamed, Ayman El-Faham, A. A. El-Bardan, and E. F. Saad “Correlation and Spectral Studies of Some Aryl Sulfides and Sulfones” in the Thirteenth of IUPAC Conference on Physical Organic Chemistry, Seoul, Korea, 1996.
- S. A. Kates, S. A. Triolo, E. Diekmann, L. A. Carpino, Ayman El-Faham, D. Ionescu, and F. Albericio “Recent Developments in Azabenzotriazole-Based Coupling Reagents for Use in Solid Phase Peptide Synthesis” in Proceeding of the Fourteenth American Peptide Symposium (Eds. P. T. Kaumaya and R. S. Hoges) Mayflower Scientific Ltd-England, 1996, pp115-116.
- H. Wenschuh, M. Beyermann, M. Bienert, Ayman El-Faham, S. Ghassemi, and L. A. Carpino “Scope and Limitations of FMOC Amino Acid Fluorides as Reagents for Peptide Synthesis” in Proceeding of the Fourteenth American Peptide Symposium (Eds. P. T. Kaumaya and R. S. Hoges) Mayflower Scientific Ltd-England, 1996, pp33-35.
- S. A. Kates, E. Diekmann, Ayman El-Faham, L. W. Herman, D. Ionescu, B. F. McGuinness, S. A. Triolo, F. Albericio, and L. A. Carpino “ On the Use of Novel Coupling Reagents for Solid Phase Peptide Synthesis”Techniques in Protein Chemistry VII, (Ed., D. R. Marsshak), Academic Press, New York, 1996, pp 515-523.
- S. A. Kates, C. A. Minor, H. Shroff, R. C. Haaseth, S. A. Triolo, Ayman El-Faham, L. A. Carpino, and F. Albericio “Practical Protocols for Efficient Solid Phase Peptide Synthesis: Minimization of Side-Reactions” in Proceeding of the Twenty-Thrid European Peptide Symposium (Ed. H. S. Maia) Escom, Leiden, The Netherland, 1995, pp 248-249.
- F. Albericio, I. Abdelmoty, J. M. Bofill, L. A. Carpino, Ayman El-Faham, B. M. Foxman, M. Gairi, E. Giralt, G. W. Griffin, S. A. Kates, P. LIoyd-Williams, C. A. Minor, L. M. Scarmoutzos, H. Shroff, S. Triolo, and H. Wenschuh “ Azabenzo- triazole (HOAt) Derivatives as Superior Coupling Reagent for Peptide Synthesis” in Proceeding the Twenty-Third European Peptide Symposium (Ed. H. L. S. Maia) Escom, Leiden, 1995, pp 23-25.
- L. A. Carpino, Ayman El-Faham, G. A. Truran, S. A. Triolo, H. Shroff, G. W. Grifin, C. A. Minor, S. A. Kates, and F. Albericio “Azabenzotriazole-Based Coupling Reagents in Solid Phase Peptide Synthesis” in Proceeding the Thirteenth American Peptide Symposium (Ed. R. S. Wodges and J. A. Smith) Escom, Leiden, 1994, pp 124-126.
- L. A. Carpino, Ayman El-Faham, G. A. Truran, C. A. Minor, S. A. Kates, G. W. Grifin, H. Shroff, S. A. Triolo, and F. Albericio “New Approaches for Extending the Scope of Solid Phase Peptide Synthesis” in Innovation and Perspective in the Solid Phase Peptide Synthesis: Peptides Proteins and Nucleic Acid, Biological and Biochemical Application (Ed. R. Epton) Mayflower Worldwide Limited, Birmingham, England, 1994, pp 95-104.
- F. Albericio. L. A. Carpino, S. B. Daniels, Ayman El-Faham, H. Fukuda, G. W. Griffin, S. A. Kates, C. A. Minor, H. N. Shroff, S. A. Triolo, G. T. Truran, and K. Yamabe “New approaches in Solid Phase Peptide Synthesis” in Proceeding of the 31th symposium on Peptide Chemistry (Ed. Y. Okada) Minoh-shi, Osaka 562, Japan, 1994, pp 121-124.